Dapsone (BioDeep_00000001703)

 

Secondary id: BioDeep_00000408881

human metabolite blood metabolite


代谢物信息卡片


4-(4-Amino-benzenesulphonyl)-phenylamine

化学式: C12H12N2O2S (248.0619452)
中文名称: 4,4-二氨基二苯砜
谱图信息: 最多检出来源 Homo sapiens(blood) 16.67%

分子结构信息

SMILES: C1=CC(=CC=C1N)S(=O)(=O)C2=CC=C(C=C2)N
InChI: InChI=1S/C12H12N2O2S/c13-9-1-5-11(6-2-9)17(15,16)12-7-3-10(14)4-8-12/h1-8H,13-14H2

描述信息

A sulfone active against a wide range of bacteria but mainly employed for its actions against mycobacterium leprae. Its mechanism of action is probably similar to that of the sulfonamides which involves inhibition of folic acid synthesis in susceptible organisms. It is also used with pyrimethamine in the treatment of malaria. (From Martindale, The Extra Pharmacopoeia, 30th ed, p157-8)
CONFIDENCE standard compound; INTERNAL_ID 857; DATASET 20200303_ENTACT_RP_MIX501; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 5725; ORIGINAL_PRECURSOR_SCAN_NO 5723
CONFIDENCE standard compound; INTERNAL_ID 857; DATASET 20200303_ENTACT_RP_MIX501; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 5706; ORIGINAL_PRECURSOR_SCAN_NO 5704
CONFIDENCE standard compound; INTERNAL_ID 857; DATASET 20200303_ENTACT_RP_MIX501; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 5675; ORIGINAL_PRECURSOR_SCAN_NO 5671
CONFIDENCE standard compound; INTERNAL_ID 857; DATASET 20200303_ENTACT_RP_MIX501; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 5709; ORIGINAL_PRECURSOR_SCAN_NO 5707
CONFIDENCE standard compound; INTERNAL_ID 857; DATASET 20200303_ENTACT_RP_MIX501; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 5694; ORIGINAL_PRECURSOR_SCAN_NO 5692
CONFIDENCE standard compound; INTERNAL_ID 857; DATASET 20200303_ENTACT_RP_MIX501; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 5720; ORIGINAL_PRECURSOR_SCAN_NO 5718
J - Antiinfectives for systemic use > J04 - Antimycobacterials > J04B - Drugs for treatment of lepra > J04BA - Drugs for treatment of lepra
D - Dermatologicals > D10 - Anti-acne preparations > D10A - Anti-acne preparations for topical use
D000890 - Anti-Infective Agents > D000977 - Antiparasitic Agents > D000981 - Antiprotozoal Agents
D000890 - Anti-Infective Agents > D000900 - Anti-Bacterial Agents > D007917 - Leprostatic Agents
COVID info from clinicaltrial, clinicaltrials, clinical trial, clinical trials
C254 - Anti-Infective Agent > C849 - Sulfone Anti-Infective Agent
D004791 - Enzyme Inhibitors > D005493 - Folic Acid Antagonists
CONFIDENCE standard compound; EAWAG_UCHEM_ID 3644
CONFIDENCE standard compound; INTERNAL_ID 1024
KEIO_ID A220; [MS2] KO008829
KEIO_ID A220
Corona-virus
Coronavirus
SARS-CoV-2
COVID-19
SARS-CoV
COVID19
SARS2
SARS

同义名列表

58 个代谢物同义名

4-(4-Amino-benzenesulphonyl)-phenylamine; 4-(4-Amino-benzenesulfonyl)-phenylamine; 4-(4-Aminophenylsulphonyl)benzenamine; 4-(4-Aminophenylsulfonyl)benzenamine; 4-(4-aminobenzenesulfonyl)aniline; 4-(4-Aminophenylsulphonyl)aniline; 1,1-Sulphonylbis(4-aminobenzene); 4-(4-Aminophenylsulfonyl)aniline; 1,1-Sulfonylbis(4-aminobenzene); 1,1-Sulfonylbis[4-aminobenzene]; Mex-america brand OF dapsone; 4,4-Diaminodiphenyl sulphone; p,P-diaminodiphenyl sulphone; p,p-Sulphonylbisbenzenamine; 4,4-Diaminodiphenyl sulfone; 4,4-Sulfonylbisbenzeneamine; Bis(p-aminophenyl) sulphone; p,P-diaminodiphenyl sulfone; 4,4-Sulphonylbisbenzenamine; Bis(4-aminophenyl)sulphone; 4,4-Sulfonylbisbenzenamine; Bis(p-aminophenyl) sulfone; Sulfone, 4,4-diaminophenyl; 4,4-Diaminodiphenylsulfone; p,p-Sulfonylbisbenzenamine; 4,4-Diaminophenyl sulfone; 4,4 Diaminophenyl sulfone; p,p-Sulphonylbisbenzamine; Bis(4-aminophenyl)sulfone; p,p-Sulfonylbisbenzamine; 4,4-Sulphonylbisaniline; Orsade brand OF dapsone; Fatol brand OF dapsone; Diaminodiphenylsulfone; p-Aminophenyl sulphone; 4-Aminophenyl sulphone; 4,4-Sulfonylbisaniline; 4,4-Sulfonyldianiline; 4-Aminophenyl sulfone; p-Aminophenyl sulfone; 4-Aminophenylsulfone; 4,4-Sulfonyldianilin; DDS, Pharmaceutical; Sulfonyldianiline; DIAPHENYLsulphone; DIAPHENYLsulfone; Dapson-fatol; 4,4-Dapsone; Avlosulfone; Dapsoderm-X; Dapsonum; Disulone; Sulfona; Dapsona; dapsone; Aczone; DADPS; DDS



数据库引用编号

47 个数据库交叉引用编号

分类词条

相关代谢途径

Reactome(0)

BioCyc(0)

PlantCyc(0)

代谢反应

0 个相关的代谢反应过程信息。

Reactome(0)

BioCyc(0)

WikiPathways(0)

Plant Reactome(0)

INOH(0)

PlantCyc(0)

COVID-19 Disease Map(0)

PathBank(0)

PharmGKB(0)

1 个相关的物种来源信息

在这里通过桑基图来展示出与当前的这个代谢物在我们的BioDeep知识库中具有相关联信息的其他代谢物。在这里进行关联的信息来源主要有：

  • PubMed: 来源于PubMed文献库中的文献信息，我们通过自然语言数据挖掘得到的在同一篇文献中被同时提及的相关代谢物列表，这个列表按照代谢物同时出现的文献数量降序排序，取前10个代谢物作为相关研究中关联性很高的代谢物集合展示在桑基图中。
  • NCBI Taxonomy: 通过文献数据挖掘，得到的代谢物物种来源信息关联。这个关联信息同样按照出现的次数降序排序，取前10个代谢物作为高关联度的代谢物集合展示在桑吉图上。
  • Chemical Taxonomy: 在物质分类上处于同一个分类集合中的其他代谢物
  • Chemical Reaction: 在化学反应过程中，存在为当前代谢物相关联的生化反应过程中的反应底物或者反应产物的关联代谢物信息。

点击图上的相关代谢物的名称，可以跳转到相关代谢物的信息页面。



文献列表

  • Thakur Rohit Singh, Devaraj Ezhilarasan. Lagerstroemia speciosa (L.) Pers., ethanolic leaves extract attenuates dapsone-induced liver inflammation in rats. Drug and chemical toxicology. 2022 Sep; 45(5):2361-2370. doi: 10.1080/01480545.2021.1945079. [PMID: 34225555]
  • Mohammad Reza Madanipour, Mortaza Fatehi-Zardalou, Nastaran Rahimi, Sara Hemmati, Mojgan Alaeddini, Shahroo Etemad-Moghadam, Maryam Shayan, Sasan Dabiri, Ahmad Reza Dehpour. The anti-inflammatory effect of dapsone on ovalbumin-induced allergic rhinitis in balb/c mice. Life sciences. 2022 May; 297(?):120449. doi: 10.1016/j.lfs.2022.120449. [PMID: 35245518]
  • G S Basavaraj, Riddhi Das Gupta, Bhavesh Patel, Felix Jebasingh, Anu Anna George, Dincy Peter, Leni George, Thomas V Paul, Nihal Thomas. Erroneous reduction of HbA1c levels in patients with type 2 diabetes mellitus on dapsone treatment for Hansen's disease - a single-center retrospective cohort study. Indian journal of dermatology, venereology and leprology. 2022 May; 88(4):519-522. doi: 10.25259/ijdvl_527_18. [PMID: 33871212]
  • Akshay Khatri, Sarath Lal M R, Madhu C Bhaskaran. Dapsone-Associated Hemolytic Anemia in Renal Transplant Recipients With Normal Glucose-6-Phosphate-Dehydrogenase Levels. American journal of therapeutics. 2022 May; 29(3):e369-e372. doi: 10.1097/mjt.0000000000001252. [PMID: 32947344]
  • Xuesong Wang, Zhenzhen Wang, Lulu Sun, Hong Liu, Furen Zhang. Efficacy and safety of dapsone gel for acne: a systematic review and meta-analysis. Annals of palliative medicine. 2022 Feb; 11(2):611-620. doi: 10.21037/apm-21-3935. [PMID: 35249339]
  • Marco Andrey Cipriani Frade, Fred Bernardes Filho, Ana Laura Quirino de Lima, Marcelo Bezerra de Menezes, Helena Barbosa Lugão. Asymptomatic low pulse oximetry measurements in leprosy patients in the time of COVID-19: Dapsone side effect. Revista da Sociedade Brasileira de Medicina Tropical. 2022; 55(?):e0491. doi: 10.1590/0037-8682-0491-2021. [PMID: 35239908]
  • Shasank Sekhar Swain, Gunanidhi Sahoo, Pravati Kumari Mahapatra, Sujogya Kumar Panda. Disease Burden and Current Therapeutical Status of Leprosy with Special Emphasis on Phytochemicals. Current topics in medicinal chemistry. 2022; 22(19):1611-1625. doi: 10.2174/1568026621666210909162435. [PMID: 34503409]
  • Samira Shirooie, Ehsan Khaledi, Ahmad Reza Dehpour, Tayebeh Noori, Mozafar Khazaei, Faezeh Sadeghi, Eduardo Sobarzo-Sánchez. The effect of dapsone in testosterone enanthate-induced polycystic ovary syndrome in rat. The Journal of steroid biochemistry and molecular biology. 2021 11; 214(?):105977. doi: 10.1016/j.jsbmb.2021.105977. [PMID: 34428594]
  • Alfonso Mata-Bermudez, Araceli Diaz-Ruiz, Masha Burelo, Betzabeth Anali García-Martínez, Gustavo Jardon-Guadarrama, Francisco Calderón-Estrella, Andrea Rangel-Hernández, Cuauhtémoc Pérez-González, Rios Camilo. Dapsone Prevents Allodynia and Hyperalgesia and Decreased Oxidative Stress After Spinal Cord Injury in Rats. Spine. 2021 Oct; 46(19):1287-1294. doi: 10.1097/brs.0000000000004015. [PMID: 34517396]
  • T Tripathi, A R Singh, R Kapoor, A Sinha, S Ghosh, K Kaur, D Pokhariya, S Maity, A Tapadar, A Chandra. Dapsone-induced methaemoglobinaemia in leprosy: a close mimic of 'happy hypoxia' in the COVID-19 pandemic. Journal of the European Academy of Dermatology and Venereology : JEADV. 2021 09; 35(9):e568-e571. doi: 10.1111/jdv.17394. [PMID: 34037283]
  • Chiara Sabbadin, Alessandra Andrisani, Gabriella Donà, Elena Tibaldi, Anna Maria Brunati, Stefano Dall'Acqua, Eugenio Ragazzi, Guido Ambrosini, Decio Armanini, Luciana Bordin. Endometriosis Susceptibility to Dapsone-Hydroxylamine-Induced Alterations Can Be Prevented by Licorice Intake: In Vivo and In Vitro Study. International journal of molecular sciences. 2021 Aug; 22(16):. doi: 10.3390/ijms22168476. [PMID: 34445180]
  • Sai Sudha Mannemuddhu, Rozina Ali, Salam Kadhem, Rupam Ruchi. Unusual cause of persistent dyspnea in a patient with nephrotic syndrome: dapsone-induced methemoglobinemia. CEN case reports. 2021 08; 10(3):336-340. doi: 10.1007/s13730-020-00565-8. [PMID: 33417185]
  • Selma Regina Penha Silva Cerqueira, Patrícia Duarte Deps, Débora Vilela Cunha, Natanael Victor Furtunato Bezerra, Daniel Holanda Barroso, Ana Bárbara Sapienza Pinheiro, Gecilmara Salviato Pillegi, Taynah Alves Rocha Repsold, Patrícia Shu Kurizky, Simon M Collin, Ciro Martins Gomes. The influence of leprosy-related clinical and epidemiological variables in the occurrence and severity of COVID-19: A prospective real-world cohort study. PLoS neglected tropical diseases. 2021 07; 15(7):e0009635. doi: 10.1371/journal.pntd.0009635. [PMID: 34319982]
  • Aditi Hindka, Dao Huynh, Priya S Verghese. Dapsone-induced methemoglobinemia in pediatrics post-renal transplant. Pediatric transplantation. 2021 May; 25(3):e13921. doi: 10.1111/petr.13921. [PMID: 33280223]
  • Mark J Henderson, Kathleen A Trychta, Shyh-Ming Yang, Susanne Bäck, Adam Yasgar, Emily S Wires, Carina Danchik, Xiaokang Yan, Hideaki Yano, Lei Shi, Kuo-Jen Wu, Amy Q Wang, Dingyin Tao, Gergely Zahoránszky-Kőhalmi, Xin Hu, Xin Xu, David Maloney, Alexey V Zakharov, Ganesha Rai, Fumihiko Urano, Mikko Airavaara, Oksana Gavrilova, Ajit Jadhav, Yun Wang, Anton Simeonov, Brandon K Harvey. A target-agnostic screen identifies approved drugs to stabilize the endoplasmic reticulum-resident proteome. Cell reports. 2021 04; 35(4):109040. doi: 10.1016/j.celrep.2021.109040. [PMID: 33910017]
  • Sriram Sriperumbuduri, Caitlin Hesketh, Edward G Clark. A Transplant Patient with Blue Lips, Tongue, and Fingertips. Kidney360. 2021 02; 2(2):398-399. doi: 10.34067/kid.0005102020. [PMID: 35373029]
  • Rita Sampaio, Leandro Silva, Goreti Catorze, Isabel Viana. Cutaneous Rosai-Dorfman disease: a challenging diagnosis. BMJ case reports. 2021 Feb; 14(2):. doi: 10.1136/bcr-2020-239244. [PMID: 33541998]
  • Sunmeet Sandhu, Shekhar Neema, Deepak Vashisht, Ruby Venugopal, Prashant Sengupta, Subramaniyan Radhakrishnan. Drug reaction with eosinophilia and systemic symptoms: A single center descriptive observational study. Dermatologic therapy. 2021 01; 34(1):e14670. doi: 10.1111/dth.14670. [PMID: 33314590]
  • Gabriela Schneider-Rauber, Debora Fretes Argenta, Thiago Caon. Emerging Technologies to Target Drug Delivery to the Skin - the Role of Crystals and Carrier-Based Systems in the Case Study of Dapsone. Pharmaceutical research. 2020 Nov; 37(12):240. doi: 10.1007/s11095-020-02951-4. [PMID: 33169237]
  • Ömer Faruk Elmas, Abdullah Demirbaş, Ümit Türsen, Mustafa Atasoy, Torello Lotti. Pemphigus and COVID-19: Critical overview of management with a focus on treatment choice. Dermatologic therapy. 2020 11; 33(6):e14265. doi: 10.1111/dth.14265. [PMID: 32882079]
  • Jong-Hoon Lee, Ha Kyeu An, Mun-Gi Sohn, Paul Kivela, Sangsuk Oh. 4,4'-Diaminodiphenyl Sulfone (DDS) as an Inflammasome Competitor. International journal of molecular sciences. 2020 Aug; 21(17):. doi: 10.3390/ijms21175953. [PMID: 32824985]
  • Eric L Altschuler, Richard E Kast. Dapsone, colchicine and olanzapine as treatment adjuncts to prevent COVID-19 associated adult respiratory distress syndrome (ARDS). Medical hypotheses. 2020 08; 141(?):109774. doi: 10.1016/j.mehy.2020.109774. [PMID: 32344275]
  • Ahmed Farouk, Samar Salman. Dapsone and doxycycline could be potential treatment modalities for COVID-19. Medical hypotheses. 2020 07; 140(?):109768. doi: 10.1016/j.mehy.2020.109768. [PMID: 32339778]
  • Joseph George. Metabolism and interactions of antileprosy drugs. Biochemical pharmacology. 2020 07; 177(?):113993. doi: 10.1016/j.bcp.2020.113993. [PMID: 32339493]
  • Sadaf Nezamoleslami, Mohammad Sheibani, Fatemeh Jahanshahi, Faiza Mumtaz, Ata Abbasi, Ahmad Reza Dehpour. Protective effect of dapsone against renal ischemia-reperfusion injury in rat. Immunopharmacology and immunotoxicology. 2020 Jun; 42(3):272-279. doi: 10.1080/08923973.2020.1755308. [PMID: 32321337]
  • Mohammad Sheibani, Sadaf Nezamoleslami, Hedyeh Faghir-Ghanesefat, Amir Hossein Emami, Ahmad Reza Dehpour. Cardioprotective effects of dapsone against doxorubicin-induced cardiotoxicity in rats. Cancer chemotherapy and pharmacology. 2020 03; 85(3):563-571. doi: 10.1007/s00280-019-04019-6. [PMID: 31915967]
  • Gurinder Kumar, Hanan Khalid AlHadhrami. Bullous lesions in a young adolescent postrenal transplant. Saudi journal of kidney diseases and transplantation : an official publication of the Saudi Center for Organ Transplantation, Saudi Arabia. 2020 Mar; 31(2):553-555. doi: 10.4103/1319-2442.284037. [PMID: 32394935]
  • Christopher Evernden, Michelle Dowhan, Rosy Dabas, Ahsan Chaudhry, Amit Kalra, Poonam Dharmani-Khan, Daniel Gregson, Andrew Johnson, Jennifer Jupp, Victor Jimenez-Zepeda, Kareem Jamani, Peter Duggan, Jason Tay, Faisal Khan, Andrew Daly, Jan Storek. High incidence of Pneumocystis jirovecii pneumonia in allogeneic hematopoietic cell transplant recipients in the modern era. Cytotherapy. 2020 01; 22(1):27-34. doi: 10.1016/j.jcyt.2019.11.002. [PMID: 31889628]
  • Mohammed Elmowafy, Khaled Shalaby, Hazim M Ali, Nabil K Alruwaili, Ayman Salama, Mohamed F Ibrahim, Mohamed A Akl, Tarek A Ahmed. Impact of nanostructured lipid carriers on dapsone delivery to the skin: in vitro and in vivo studies. International journal of pharmaceutics. 2019 Dec; 572(?):118781. doi: 10.1016/j.ijpharm.2019.118781. [PMID: 31715347]
  • Rohini Kanwar, Michael Gradzielski, Sylvain Prevost, Gurpreet Kaur, Marie-Sousai Appavou, S K Mehta. Physicochemical stimuli as tuning parameters to modulate the structure and stability of nanostructured lipid carriers and release kinetics of encapsulated antileprosy drugs. Journal of materials chemistry. B. 2019 11; 7(42):6539-6555. doi: 10.1039/c9tb01330j. [PMID: 31584603]
  • Tobie D Lee, Olivia W Lee, Kyle R Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G Tebase, Carleen Klumpp-Thomas, Robert W Robey, Suresh V Ambudkar, Min Shen, Michael M Gottesman, Matthew D Hall. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. Molecular pharmacology. 2019 11; 96(5):629-640. doi: 10.1124/mol.119.115964. [PMID: 31515284]
  • Julia Torabi, Alesa Campbell, Gayatri Nair, Gauravkumar L Patel, Yoshifumi Miura, Jay A Graham. Dapsone-Induced Methemoglobinemia in Two Renal Transplant Recipients. Progress in transplantation (Aliso Viejo, Calif.). 2019 09; 29(3):289-290. doi: 10.1177/1526924819855365. [PMID: 31167609]
  • Céline Roman, Bogdan Dima, Laurence Muyshont, Thierry Schurmans, Olivier Gilliaux. Indications and efficiency of dapsone in IgA vasculitis (Henoch-Schonlein purpura): case series and a review of the literature. European journal of pediatrics. 2019 Aug; 178(8):1275-1281. doi: 10.1007/s00431-019-03409-5. [PMID: 31230197]
  • Sherrie J Divito. Screening HLA to Prevent Severe Drug Reactions-A Devil's Advocate Perspective. JAMA dermatology. 2019 06; 155(6):655-656. doi: 10.1001/jamadermatol.2018.5336. [PMID: 30916720]
  • Ekta Varshney, Monika Tandon, Nilanjan Saha, Shakir Ali. In vivo phenotyping of cytochrome 450 isoforms involved in the metabolism of anti-HIV and anti-tubercular drugs in human using cocktail approach: An LC-MS/MS analysis. Journal of pharmaceutical and biomedical analysis. 2019 Feb; 164(?):698-705. doi: 10.1016/j.jpba.2018.11.026. [PMID: 30472588]
  • Yuri de Deus Mont'alverne Parente, Amanda Lopes de Castro, Flávio Bezerra de Araújo, André Costa Teixeira, Ítalo Criszostomo Lima, Elizabeth De Francesco Daher. Acute renal failure by rapidly progressive glomerulonephritis with IgA deposition in a patient concomitantly diagnosed with multibacillary Hansen's disease: a case report. Jornal brasileiro de nefrologia : 'orgao oficial de Sociedades Brasileira e Latino-Americana de Nefrologia. 2019 Jan; 41(1):152-156. doi: 10.1590/2175-8239-jbn-2018-0056. [PMID: 30160772]
  • Franziska Hübner, Michael Kasperkiewicz, Diana Knuth-Rehr, Iakov Shimanovich, Joachim Hübner, Sven Süfke, Philip Muck, Detlef Zillikens, Enno Schmidt. Adjuvant treatment of severe/refractory bullous pemphigoid with protein A immunoadsorption. Journal der Deutschen Dermatologischen Gesellschaft = Journal of the German Society of Dermatology : JDDG. 2018 Sep; 16(9):1109-1118. doi: 10.1111/ddg.13642. [PMID: 30179319]
  • Emma F Johnson, Stanislav N Tolkachjov, Lawrence E Gibson. Alpha-1 antitrypsin deficiency panniculitis: clinical and pathologic characteristics of 10 cases. International journal of dermatology. 2018 Aug; 57(8):952-958. doi: 10.1111/ijd.14012. [PMID: 29707779]
  • Rohini Kanwar, Michael Gradzielski, S K Mehta. Biomimetic Solid Lipid Nanoparticles of Sophorolipids Designed for Antileprosy Drugs. The journal of physical chemistry. B. 2018 07; 122(26):6837-6845. doi: 10.1021/acs.jpcb.8b03081. [PMID: 29874078]
  • Wei-Ti Chen, Chuang-Wei Wang, Chun-Wei Lu, Chun-Bing Chen, Hua-En Lee, Shuen-Iu Hung, Siew-Eng Choon, Chih-Hsun Yang, Ming-Tsan Liu, Ting Jui Chen, Wen-Lang Fan, Shih-Chi Su, Yang Yu-Wei Lin, Ya-Ching Chang, Wen-Hung Chung. The Function of HLA-B*13:01 Involved in the Pathomechanism of Dapsone-Induced Severe Cutaneous Adverse Reactions. The Journal of investigative dermatology. 2018 07; 138(7):1546-1554. doi: 10.1016/j.jid.2018.02.004. [PMID: 29458119]
  • Rui Zhan, Mingming Zhao, Ting Zhou, Yue Chen, Weiwei Yu, Lei Zhao, Tao Zhang, Hecheng Wang, Huan Yang, Yinglan Jin, Qihua He, Xiaoda Yang, Xiangyang Guo, Belinda Willard, Bing Pan, Yining Huang, Yingyu Chen, Dehua Chui, Lemin Zheng. Dapsone protects brain microvascular integrity from high-fat diet induced LDL oxidation. Cell death & disease. 2018 06; 9(6):683. doi: 10.1038/s41419-018-0739-y. [PMID: 29880899]
  • Hendra Gunawan, Muljaningsih Sasmojo, Helena Eka Putri, Erda Avriyanti, Reti Hindritiani, Oki Suwarsa. Clinical pilot study: Clarithromycin efficacy in multibacillary leprosy therapy. International journal of mycobacteriology. 2018 Apr; 7(2):152-155. doi: 10.4103/ijmy.ijmy_58_18. [PMID: 29900892]
  • Sanjeevani Shekhar Deshkar, Shyam Gangadhar Bhalerao, Monali Shivaji Jadhav, Satish Vasudeo Shirolkar. Formulation and Optimization of Topical Solid Lipid Nanoparticles based Gel of Dapsone Using Design of Experiment. Pharmaceutical nanotechnology. 2018; 6(4):264-275. doi: 10.2174/2211738506666181105141522. [PMID: 30394227]
  • M Sticherling, A Franke, E Aberer, R Gläser, M Hertl, C Pfeiffer, B Rzany, S Schneider, I Shimanovich, T Werfel, A Wilczek, D Zillikens, E Schmidt. An open, multicentre, randomized clinical study in patients with bullous pemphigoid comparing methylprednisolone and azathioprine with methylprednisolone and dapsone. The British journal of dermatology. 2017 Nov; 177(5):1299-1305. doi: 10.1111/bjd.15649. [PMID: 28494097]
  • Keum Hwa Lee, Jae Hyon Park, Dong Hyun Kim, Jimin Hwang, Goeun Lee, Jae Seok Hyun, Sung Taik Heo, Ji Hoon Choi, Minwoo Kim, Minhye Kim, Seong Il Kim, Michael Eisenhut, Andreas Kronbichler, Jae Il Shin. Dapsone as a potential treatment option for Henoch-Schönlein Purpura (HSP). Medical hypotheses. 2017 Oct; 108(?):42-45. doi: 10.1016/j.mehy.2017.07.018. [PMID: 29055398]
  • Sohail Abdul Salim, Lakshmi Ramachandran Nair, Venkataraman Palabindala, Iasmina Craici. Upward trend of dapsone-induced methemoglobinemia in renal transplant community
. Clinical nephrology. 2017 Sep; 88(9):156-161. doi: 10.5414/cn109181. [PMID: 28699887]
  • Coralie Lheure, Saskia Ingen-Housz-Oro, Sandra Guignard, Rachida Inaoui, Brigitte Jolivet, Xavier Chevalier, Pierre Wolkenstein, Bruno Fautrel, Oliver Chosidow. Dermatitis herpetiformis and bone mineral density: analysis of a French cohort of 53 patients. European journal of dermatology : EJD. 2017 Aug; 27(4):353-358. doi: 10.1684/ejd.2017.3029. [PMID: 28524056]
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