Chemical Formula: C10H12N2O4

Chemical Formula C10H12N2O4

Found 54 metabolite its formula value is C10H12N2O4

3-Hydroxyl kyneurenine

2-Amino-4-(2-amino-3-hydroxyphenyl)-4-oxobutanoic acid

C10H12N2O4 (224.0797032)


Hydroxykynurenine is a free radical generator and a bioprecursor quinolinic acid which is a endogenous excitotoxin (PMID 16697652). It is a product of enzyme kynurenine 3-monooxygenase in the tryptophan catabolism pathway (Reactome http://www.reactome.org). [HMDB] Hydroxykynurenine is a free radical generator and a bioprecursor quinolinic acid which is a endogenous excitotoxin (PMID 16697652). It is a product of enzyme kynurenine 3-monooxygenase in the tryptophan catabolism pathway (Reactome http://www.reactome.org). Acquisition and generation of the data is financially supported in part by CREST/JST. [Raw Data] CBA12_3-OH-kynurenine_pos_20eV_1-4_01_802.txt [Raw Data] CBA12_3-OH-kynurenine_pos_10eV_1-4_01_801.txt [Raw Data] CBA12_3-OH-kynurenine_pos_50eV_1-4_01_805.txt [Raw Data] CBA12_3-OH-kynurenine_pos_40eV_1-4_01_804.txt [Raw Data] CBA12_3-OH-kynurenine_pos_30eV_1-4_01_803.txt C26170 - Protective Agent > C275 - Antioxidant KEIO_ID H050; [MS3] KO009001 KEIO_ID H050; [MS2] KO009000 KEIO_ID H050

   

Stavudine

1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione

C10H12N2O4 (224.07970319999998)


Stavudine is only found in individuals that have used or taken this drug. It is a dideoxynucleoside analog that inhibits reverse transcriptase and has in vitro activity against HIV. [PubChem]Stavudine inhibits the activity of HIV-1 reverse transcriptase (RT) both by competing with the natural substrate dGTP and by its incorporation into viral DNA. J - Antiinfectives for systemic use > J05 - Antivirals for systemic use > J05A - Direct acting antivirals > J05AF - Nucleoside and nucleotide reverse transcriptase inhibitors C471 - Enzyme Inhibitor > C1589 - Reverse Transcriptase Inhibitor > C97452 - Nucleoside Reverse Transcriptase Inhibitor D000890 - Anti-Infective Agents > D000998 - Antiviral Agents > D018894 - Reverse Transcriptase Inhibitors D000890 - Anti-Infective Agents > D000998 - Antiviral Agents > D044966 - Anti-Retroviral Agents D009676 - Noxae > D000963 - Antimetabolites > D015224 - Dideoxynucleosides D004791 - Enzyme Inhibitors > D019384 - Nucleic Acid Synthesis Inhibitors C254 - Anti-Infective Agent > C281 - Antiviral Agent Stavudine (d4T) is an orally active nucleoside reverse transcriptase inhibitor (NRTI). Stavudine has activity against HIV-1 and HIV-2. Stavudine also inhibits the replication of mitochondrial DNA (mtDNA). Stavudine reduces NLRP3 inflammasome activation and modulates Amyloid-β autophagy. Stavudine induces apoptosis[1][2][3][4].

   

5-Hydroxykynurenine

2-Amino-4-(2-amino-5-hydroxyphenyl)-4-oxobutanoic acid

C10H12N2O4 (224.07970319999998)


5-Hydroxykynurenine is found in the tryptophan metabolism pathway. It is created from 5-Hydroxy-N-formylkynurenine through the action of arylformamidase [EC:3.5.1.9]. 5-Hydroxykynurenine is then converted to 5-Hydroxykynurenamine by the action of dopa decarboxylase [EC:4.1.1.28]. [HMDB] 5-Hydroxykynurenine is found in the tryptophan metabolism pathway. It is created from 5-Hydroxy-N-formylkynurenine through the action of arylformamidase [EC:3.5.1.9]. 5-Hydroxykynurenine is then converted to 5-Hydroxykynurenamine by the action of dopa decarboxylase [EC:4.1.1.28].

   

L-3-Hydroxykynurenine

(2S)-2-Amino-4-(2-amino-3-hydroxyphenyl)-4-oxobutanoic acid

C10H12N2O4 (224.07970319999998)


L-3-Hydroxykynurenine (L-3-HK) is a metabolite in the kynurenine pathway, the major route of tryptophan degradation in mammals. Kynurenine 3-monooxygenase, an NADPH-dependent flavin monooxygenase, catalyses the hydroxylation of L-kynurenine to L-3-hydroxykynurenine. 3-hydroxykynurenine can be converted to 3-hydroxyanthranilate by the enzyme 3-hydroxykinureninase. It may also be converted to 4-(2-amino-3-hydroxphenyl)-2,4-dioxobutanoate by the enzyme kynurenine-oxoglutarate transaminase. L-3-Hydroxykynurenine (L-3-HK) is a known generator of highly reactive free radicals. An elevation of L-3-HK levels has been shown to constitute a significant hazard in situations of excitotoxic injury. In particular, L-3-HK may contribute to the neuronal deficits underlying HIV-associated dementia (PMID: 7830088). Pharmacological interventions aimed at decreasing L-3-HK formation may therefore be particularly useful for the treatment of neurological diseases which are associated with an abnormally enhanced flux through the kynurenine pathway (PMID: 10583474) [HMDB] L-3-Hydroxykynurenine (L-3-HK) is a metabolite in the kynurenine pathway, the major route of tryptophan degradation in mammals. Kynurenine 3-monooxygenase, an NADPH-dependent flavin monooxygenase, catalyses the hydroxylation of L-kynurenine to L-3-hydroxykynurenine. 3-hydroxykynurenine can be converted to 3-hydroxyanthranilate by the enzyme 3-hydroxykinureninase. It may also be converted to 4-(2-amino-3-hydroxphenyl)-2,4-dioxobutanoate by the enzyme kynurenine-oxoglutarate transaminase. L-3-Hydroxykynurenine (L-3-HK) is a known generator of highly reactive free radicals. An elevation of L-3-HK levels has been shown to constitute a significant hazard in situations of excitotoxic injury. In particular, L-3-HK may contribute to the neuronal deficits underlying HIV-associated dementia (PMID: 7830088). Pharmacological interventions aimed at decreasing L-3-HK formation may therefore be particularly useful for the treatment of neurological diseases which are associated with an abnormally enhanced flux through the kynurenine pathway (PMID: 10583474).

   

L-Nicotianine

1-(3-amino-3-carboxypropyl)pyridin-1-ium-3-carboxylate

C10H12N2O4 (224.07970319999998)


L-Nicotianine is found in mushrooms. L-Nicotianine is a constituent of Lentinus edodes (shiitake)

   

3-Hydroxykynurenine

3-hydroxy-dl-kynurenine

C10H12N2O4 (224.07970319999998)


A hydroxykynurenine that is kynurenine substituted by a hydroxy group at position 3. C26170 - Protective Agent > C275 - Antioxidant MS2 deconvoluted using MS2Dec from all ion fragmentation data, MetaboLights identifier MTBLS1040; VCKPUUFAIGNJHC-UHFFFAOYSA-N_STSL_0007_3-Hydroxy-DL-Kynurenine_8000fmol_180416_S2_LC02_MS02_13; Spectrum acquired as described in Naz et al 2017 PMID 28641411. Preparation and submission to MassBank of North America by Chaleckis R. and Tada I. MS2 deconvoluted using CorrDec from all ion fragmentation data, MetaboLights identifier MTBLS1040; Spectrum acquired as described in Naz et al 2017 PMID 28641411. Preparation and submission to MassBank of North America by Chaleckis R. and Tada I.

   
   
   
   

Stavudine

Stavudine

C10H12N2O4 (224.07970319999998)


J - Antiinfectives for systemic use > J05 - Antivirals for systemic use > J05A - Direct acting antivirals > J05AF - Nucleoside and nucleotide reverse transcriptase inhibitors C471 - Enzyme Inhibitor > C1589 - Reverse Transcriptase Inhibitor > C97452 - Nucleoside Reverse Transcriptase Inhibitor D000890 - Anti-Infective Agents > D000998 - Antiviral Agents > D018894 - Reverse Transcriptase Inhibitors D000890 - Anti-Infective Agents > D000998 - Antiviral Agents > D044966 - Anti-Retroviral Agents D009676 - Noxae > D000963 - Antimetabolites > D015224 - Dideoxynucleosides D004791 - Enzyme Inhibitors > D019384 - Nucleic Acid Synthesis Inhibitors C254 - Anti-Infective Agent > C281 - Antiviral Agent CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 2238; ORIGINAL_PRECURSOR_SCAN_NO 2235 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 2232; ORIGINAL_PRECURSOR_SCAN_NO 2230 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 2236; ORIGINAL_PRECURSOR_SCAN_NO 2234 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 2225; ORIGINAL_PRECURSOR_SCAN_NO 2224 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 2291; ORIGINAL_PRECURSOR_SCAN_NO 2290 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 2235; ORIGINAL_PRECURSOR_SCAN_NO 2233 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX503; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 9439; ORIGINAL_PRECURSOR_SCAN_NO 9434 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX503; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 9398; ORIGINAL_PRECURSOR_SCAN_NO 9395 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 9567; ORIGINAL_PRECURSOR_SCAN_NO 9562 CONFIDENCE standard compound; INTERNAL_ID 1066; DATASET 20200303_ENTACT_RP_MIX505; DATA_PROCESSING MERGING RMBmix ver. 0.2.7; DATA_PROCESSING PRESCREENING Shinyscreen ver. 0.8.0; ORIGINAL_ACQUISITION_NO 9454; ORIGINAL_PRECURSOR_SCAN_NO 9450 Stavudine (d4T) is an orally active nucleoside reverse transcriptase inhibitor (NRTI). Stavudine has activity against HIV-1 and HIV-2. Stavudine also inhibits the replication of mitochondrial DNA (mtDNA). Stavudine reduces NLRP3 inflammasome activation and modulates Amyloid-β autophagy. Stavudine induces apoptosis[1][2][3][4].

   
   
   
   
   

L-Nicotianine

1-(3-amino-3-carboxypropyl)pyridin-1-ium-3-carboxylate

C10H12N2O4 (224.07970319999998)


   

methyl 3-(ethylamino)-4-nitrobenzoate

methyl 3-(ethylamino)-4-nitrobenzoate

C10H12N2O4 (224.07970319999998)


   
   
   
   

4,6-DIAMINO-1,3-BENZENEDICARBOXYLIC ACID DIMETHYL ESTER

4,6-DIAMINO-1,3-BENZENEDICARBOXYLIC ACID DIMETHYL ESTER

C10H12N2O4 (224.07970319999998)


   

methyl 4-(ethylamino)-3-nitrobenzoate

methyl 4-(ethylamino)-3-nitrobenzoate

C10H12N2O4 (224.07970319999998)


   

2-(1,3-benzodioxol-5-yloxy)propanehydrazide

2-(1,3-benzodioxol-5-yloxy)propanehydrazide

C10H12N2O4 (224.07970319999998)


   
   

N-(4-Nitrophenyl)-2-hydroxy-2-methylpropanamide

N-(4-Nitrophenyl)-2-hydroxy-2-methylpropanamide

C10H12N2O4 (224.07970319999998)


   
   

Benzene,1,2,3,4-tetramethyl-5,6-dinitro-

Benzene,1,2,3,4-tetramethyl-5,6-dinitro-

C10H12N2O4 (224.07970319999998)


   

methyl 2-[(3-amino-2-hydroxy-benzoyl)amino]acetate

methyl 2-[(3-amino-2-hydroxy-benzoyl)amino]acetate

C10H12N2O4 (224.07970319999998)


   

4-(1-oxidopyridin-4-ylidene)pyridin-1-ium 1-oxide,hydrate

4-(1-oxidopyridin-4-ylidene)pyridin-1-ium 1-oxide,hydrate

C10H12N2O4 (224.07970319999998)


   

N-ETHOXYCARBONYL-5-NITRO-O-TOLUIDINE

N-ETHOXYCARBONYL-5-NITRO-O-TOLUIDINE

C10H12N2O4 (224.07970319999998)


   

ethyl N-(4-methyl-3-nitrophenyl)carbamate

ethyl N-(4-methyl-3-nitrophenyl)carbamate

C10H12N2O4 (224.07970319999998)


   

N-ETHOXYCARBONYL-3-NITRO-O-TOLUIDINE

N-ETHOXYCARBONYL-3-NITRO-O-TOLUIDINE

C10H12N2O4 (224.07970319999998)


   
   

(R)-3-AMINO-4-(4-BROMOPHENYL)BUTANOICACIDHYDROCHLORIDE

(R)-3-AMINO-4-(4-BROMOPHENYL)BUTANOICACIDHYDROCHLORIDE

C10H12N2O4 (224.07970319999998)


   
   
   

4-[(2-NITROPHENYL)AMINO]BUTANOIC ACID

4-[(2-NITROPHENYL)AMINO]BUTANOIC ACID

C10H12N2O4 (224.07970319999998)


   

Ethyl 4-(methylamino)-3-nitrobenzoate

Ethyl 4-(methylamino)-3-nitrobenzoate

C10H12N2O4 (224.07970319999998)


   

4-(Isopropylamino)-3-nitrobenzoic acid

4-(Isopropylamino)-3-nitrobenzoic acid

C10H12N2O4 (224.07970319999998)


   

N-(4-Methoxy-2-methyl-5-nitrophenyl)acetamide

N-(4-Methoxy-2-methyl-5-nitrophenyl)acetamide

C10H12N2O4 (224.07970319999998)


   

(R)-2-Amino-4-(2-amino-3-hydroxyphenyl)-4-oxobutanoic acid

(R)-2-Amino-4-(2-amino-3-hydroxyphenyl)-4-oxobutanoic acid

C10H12N2O4 (224.07970319999998)


   

Methyl 2-amino-3-(4-nitrophenyl)propanoate

Methyl 2-amino-3-(4-nitrophenyl)propanoate

C10H12N2O4 (224.07970319999998)


   

L-[(N-Hydroxyamino)carbonyl]phenylalanine

L-[(N-Hydroxyamino)carbonyl]phenylalanine

C10H12N2O4 (224.07970319999998)


   

d-[(n-Hydroxyamino)carbonyl]phenylalanine

d-[(n-Hydroxyamino)carbonyl]phenylalanine

C10H12N2O4 (224.07970319999998)


   

3-Hydroxy-kynurenine

3-Hydroxy-kynurenine

C10H12N2O4 (224.07970319999998)


COVID info from COVID-19 Disease Map Corona-virus Coronavirus SARS-CoV-2 COVID-19 SARS-CoV COVID19 SARS2 SARS

   
   

(2S,3R)-4-(2-aminophenyl)-2-amino-3-hydroxy-4-oxobutanoate

(2S,3R)-4-(2-aminophenyl)-2-amino-3-hydroxy-4-oxobutanoate

C10H12N2O4 (224.07970319999998)


   

(2S,3R)-2-amino-4-(2-aminophenyl)-3-hydroxy-4-oxobutanoic acid

(2S,3R)-2-amino-4-(2-aminophenyl)-3-hydroxy-4-oxobutanoic acid

C10H12N2O4 (224.07970319999998)


   

5-hydroxy-L-kynurenine zwitterion

5-hydroxy-L-kynurenine zwitterion

C10H12N2O4 (224.07970319999998)


Tha amino acid zwitterion formed from 5-hydroxy-L-kynurenine by transfer of a proton from the carboxy to the amino group; principal microspecies at pH 7.3.

   
   

3-hydroxy-L-kynurenine zwitterion

3-hydroxy-L-kynurenine zwitterion

C10H12N2O4 (224.07970319999998)


Zwitterionic form of 3-hydroxy-L-kynurenine arising from transfer of a proton from the carboxy to the amino group; major species at pH 7.3

   

5-Hydroxykynurenine

5-Hydroxykynurenine

C10H12N2O4 (224.07970319999998)


A hydroxykynurenine that is kynurenine bearing a hydroxy group at the position 5.

   

nitroso[(2,4,5-trimethoxyphenyl)methylidene]amine

nitroso[(2,4,5-trimethoxyphenyl)methylidene]amine

C10H12N2O4 (224.07970319999998)