Chemical Formula: C33H39N7O2
Chemical Formula C33H39N7O2
Found 1 metabolite its formula value is C33H39N7O2
MRTX-1257
MRTX-1257
MRTX-1257 is a selective, irreversible, covalent and orally active KRAS G12C inhibitor, with an IC50 of 900 pM for KRAS dependent ERK phosphorylation in H358 cells[1].