Chemical Formula: C30H31FN4O2

Chemical Formula C30H31FN4O2

Found 1 metabolite its formula value is C30H31FN4O2

Mutant IDH1-IN-1

Mutant IDH1-IN-1

C30H31FN4O2 (498.2431)


Mutant IDH1-IN-1 is a mutant-selective IDH1 inhibitor with with IC50s of 4, 42, 80 and 143 nM against mutant IDH1 R132C/R132C, IDH1 R132H/R132H, IDH1 R132H/WT and wild type IDH1, respectively.