Chemical Formula: C26H24F3N7O3Se
Chemical Formula C26H24F3N7O3Se
Found 1 metabolite its formula value is C26H24F3N7O3Se
Glutaminase-IN-1
Glutaminase-IN-1
Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.