Chemical Formula: C26H24F3N7O3Se

Chemical Formula C26H24F3N7O3Se

Found 1 metabolite its formula value is C26H24F3N7O3Se

Glutaminase-IN-1

Glutaminase-IN-1

C26H24F3N7O3Se (619.105784)


Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.