Chemical Formula: C24H31Cl2N3O3

Chemical Formula C24H31Cl2N3O3

Found 1 metabolite its formula value is C24H31Cl2N3O3

ARC 239 (dihydrochloride)

ARC 239 (dihydrochloride)

C24H31Cl2N3O3 (479.1742356)


ARC 239 dihydrochloride is a selective α2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at α2A, α2B, and α2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively[1].