Chemical Formula: C19H27ClF2N2O2

Chemical Formula C19H27ClF2N2O2

Found 1 metabolite its formula value is C19H27ClF2N2O2

EST73502 (monohydrochloride)

EST73502 (monohydrochloride)

C19H27ClF2N2O2 (388.1729)


EST73502 monohydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 monohydrochloride has antinociceptive activity[1].