Chemical Formula: C18H21Cl3N4O

Chemical Formula C18H21Cl3N4O

Found 1 metabolite its formula value is C18H21Cl3N4O

Clozapine N-oxide (dihydrochloride)

Clozapine N-oxide (dihydrochloride)

C18H21Cl3N4O (414.0780866)


Clozapine N-oxide dihydrochloride is a major metabolite of Clozapine and a human muscarinic designer receptors (DREADDs) agonist. Clozapine N-oxide dihydrochloride activates the DREADD receptor hM3Dq and hM4Di. Clozapine N-oxide dihydrochloride can cross the blood-brain barrier[1][2][3][4]. Clozapine is a potent dopamine antagonist and also a potent and selective muscarinic M4 receptor (EC50=11 nM) agonist[5][6].