Chemical Formula: C16H25ClN4O2
Chemical Formula C16H25ClN4O2
Found 4 metabolite its formula value is C16H25ClN4O2
(1R,4R)-[4-(4-Chloro-5-Methyl-pyriMidin-2-ylaMino)-cyclohexyl]-carbaMic acid tert-butyl ester
(1R,4R)-[4-(4-Chloro-5-Methyl-pyriMidin-2-ylaMino)-cyclohexyl]-carbaMic acid tert-butyl ester
[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester
[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester
[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester
[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester
Tracazolate (hydrochloride)
Tracazolate (hydrochloride)
Tracazolate (ICI 136753) hydrochloride is a potent GABAA receptor modulator. Tracazolate hydrochloride has selectivity for β3 and potentiates α1β1γ2s (EC50=13.2 μM), α1β3γ2 (EC50=1.5 μM). Tracazolate hydrochloride has the potency (EC50) determined by the nature of the third subunit (γ1-3, δ, ε) within the receptor complex. Tracazolate hydrochloride possesses anxiolytic and anticonvulsant activity[1][2].