Chemical Formula: C16H15BrClNO3S2

Chemical Formula C16H15BrClNO3S2

Found 1 metabolite its formula value is C16H15BrClNO3S2

BMS-986122

BMS-986122

C16H15BrClNO3S2 (446.936521)


BMS-986122 is a selective, potent positive allosteric modulator of the mu-opioid receptor (μ-OR). BMS-986122 shows potentiation of orthosteric agonist-mediated β-arrestin recruitment, adenylyl cyclase inhibition, and G protein activation. BMS-986122 potentiates DAMGO-mediated [35S]GTPγS binding in mouse brain membranes[1][2].