Exact Mass: 486.2148
Exact Mass Matches: 486.2148
Found 5 metabolites which its exact mass value is equals to given mass value 486.2148,
within given mass tolerance error 0.001 dalton. Try search metabolite list with more accurate mass tolerance error
0.0002 dalton.
N^a-Boc-N^w-(4-Methoxy-2,3,6-triMethylphenylsulfonyl)-D-arginine
N^a-Boc-N^w-(4-Methoxy-2,3,6-triMethylphenylsulfonyl)-D-arginine
4-Ethoxycarbonyl-3-[3-(ethylamino)-6-ethylimino-2,7-dimethylxanthen-9-yl]benzoic acid
4-Ethoxycarbonyl-3-[3-(ethylamino)-6-ethylimino-2,7-dimethylxanthen-9-yl]benzoic acid
TAN-452
TAN-452
TAN-452 is an orally active, selective peripherally acting δ-opioid receptor (DOR) antagonist with a Ki of 0.47?nM and a Kb of 0.21?nM. TAN-452 is an antagonist for μ-opioid receptor (MOR; Ki=36.56?nM and Kb=9.43?nM) and κ-opioid receptor (KOR; Ki=5.31?nM and Kb=7.18?nM). TAN-452, a derivative of Naltrindole, demonstrates low brain penetrability and attenuates morphine-induced side effects without affecting pain control[1].
1-[(2s,5s)-4-benzoyl-2-benzyl-5-[(7-methoxy-2h-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl]ethanone
1-[(2s,5s)-4-benzoyl-2-benzyl-5-[(7-methoxy-2h-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl]ethanone
