Exact Mass: 462.1095

Exact Mass Matches: 462.1095

Found 2 metabolites which its exact mass value is equals to given mass value 462.1095, within given mass tolerance error 0.0002 dalton. Try search metabolite list with more accurate mass tolerance error 4.0E-5 dalton.

BMS-908662 free base

BMS-908662 free base

C24H19ClN4O4 (462.1095)


   

RLX-33

RLX-33

C24H19ClN4O4 (462.1095)


RLX-33 is a potent, selective and blood-brain barrier (BBB) penetrant relaxin family peptide 3 (RXFP3) antagonist, also blocks relaxin-3-induced ERK1/2 phosphorylation, with IC50 values of 2.36 μM for RXFP3, 7.82 and 13.86 μM for ERK1 and ERK2 phosphorylation, respectively. RLX-33 can block the stimulation of food intake induced by the RXFP3-selective agonist R3/I5 in rats. RLX-33 can be used for the research of metabolic syndrome[1].