Tetraxetan (BioDeep_00000858873)
代谢物信息卡片
Tetraxetan
化学式: C16H28N4O8 (404.1907048)
中文名称: 轮环藤宁四乙酸
谱图信息:
最多检出来源 () 0%
分子结构信息
SMILES: C1CN(CCN(CCN(CCN1CC(=O)O)CC(=O)O)CC(=O)O)CC(=O)O
InChI: InChI=1S/C16H28N4O8/c21-13(22)9-17-1-2-18(10-14(23)24)5-6-20(12-16(27)28)8-7-19(4-3-17)11-15(25)26/h1-12H2,(H,21,22)(H,23,24)(H,25,26)(H,27,28)
数据库引用编号
5 个数据库交叉引用编号
- ChEBI: CHEBI:61028
- KEGGdrug: D06092
- PubChem: 121841
- ChEMBL: CHEMBL1721515
- CAS: 60239-18-1
分类词条
相关代谢途径
Reactome(0)
BioCyc(0)
PlantCyc(0)
代谢反应
0 个相关的代谢反应过程信息。
Reactome(0)
BioCyc(0)
WikiPathways(0)
Plant Reactome(0)
INOH(0)
PlantCyc(0)
COVID-19 Disease Map(0)
PathBank(0)
PharmGKB(0)
0 个相关的物种来源信息
在这里通过桑基图来展示出与当前的这个代谢物在我们的BioDeep知识库中具有相关联信息的其他代谢物。在这里进行关联的信息来源主要有：
- PubMed: 来源于PubMed文献库中的文献信息，我们通过自然语言数据挖掘得到的在同一篇文献中被同时提及的相关代谢物列表，这个列表按照代谢物同时出现的文献数量降序排序，取前10个代谢物作为相关研究中关联性很高的代谢物集合展示在桑基图中。
- NCBI Taxonomy: 通过文献数据挖掘，得到的代谢物物种来源信息关联。这个关联信息同样按照出现的次数降序排序，取前10个代谢物作为高关联度的代谢物集合展示在桑吉图上。
- Chemical Taxonomy: 在物质分类上处于同一个分类集合中的其他代谢物
- Chemical Reaction: 在化学反应过程中，存在为当前代谢物相关联的生化反应过程中的反应底物或者反应产物的关联代谢物信息。
点击图上的相关代谢物的名称，可以跳转到相关代谢物的信息页面。
文献列表
- Peipei Wang, Chen Li, Guozhu Hou, Zhaohui Li, Hongli Jing, Wen Zhang, Fang Li. Comparison of 68Ga-DOTA-FAPI-04 and 18F-FDG PET/CT in Patients With SAPHO Syndrome.
Clinical nuclear medicine.
2023 Sep; 48(9):781-784. doi:
10.1097/rlu.0000000000004724. [PMID: 37543757] - S A Sahafi-Pour, S P Shirmardi, E Saeedzadeh, S Baradaran, M Sadeghi. Internal dosimetry studies of 177Lu-BBN-GABA-DOTA, as a cancer therapy agent, in human tissues based on animal data.
Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
2022 Aug; 186(?):110273. doi:
10.1016/j.apradiso.2022.110273. [PMID: 35594697] - Sreeja Raj Menon, Arpit Mitra, Avik Chakraborty, Megha Tawate, Sudeep Sahu, Sutapa Rakshit, Sujay Gaikwad, Geetanjali Dhotre, Archana Damle, Sharmila Banerjee. Clinical Dose Preparation of [177Lu]Lu-DOTA-Pertuzumab Using Medium Specific Activity [177Lu]LuCl3 for Radioimmunotherapy of Breast and Epithelial Ovarian Cancers, with HER2 Receptor Overexpression.
Cancer biotherapy & radiopharmaceuticals.
2022 Jun; 37(5):384-402. doi:
10.1089/cbr.2021.0230. [PMID: 35575711] - Saeideh Ataei-Nakhaei, Kamran Aryana, Sayyed Mostafa Mostafavi, Hadis Mohammadzadeh Kosari, Mohammad Esmatinia, Atena Aghaee. Peptide receptor radionuclide therapy (PRRT) in radioiodine-refractory thyroid cancer: A case report of significant response to lu177 DOTA-TATE treatment.
Archives of endocrinology and metabolism.
2022 Apr; 66(2):269-271. doi:
10.20945/2359-3997000000451. [PMID: 35315988] - Hanxiang Liu, Mei Hu, Jia Deng, Yan Zhao, Dengsai Peng, Yue Feng, Li Wang, Yue Chen, Lin Qiu. A Novel Small Cyclic Peptide-Based 68Ga-Radiotracer for Positron Emission Tomography Imaging of PD-L1 Expression in Tumors.
Molecular pharmaceutics.
2022 01; 19(1):138-147. doi:
10.1021/acs.molpharmaceut.1c00694. [PMID: 34910492] - Eric J Meester, Boudewijn J Krenning, Erik de Blois, Marion de Jong, Antonius F W van der Steen, Monique R Bernsen, Kim van der Heiden. Imaging inflammation in atherosclerotic plaques, targeting SST2 with [111In]In-DOTA-JR11.
Journal of nuclear cardiology : official publication of the American Society of Nuclear Cardiology.
2021 12; 28(6):2506-2513. doi:
10.1007/s12350-020-02046-y. [PMID: 32026330] - Jasleen Kaur, Karim Arroub, Alexander Drzezga, Klaus Schomäcker, Sanjay Mathur. Synthesis, proteolytic stability, and in vitro evaluation of DOTA conjugated p160 peptide based radioconjugates: [177Lu]Lu-DOTA-p160.
Organic & biomolecular chemistry.
2021 11; 19(45):9849-9854. doi:
10.1039/d1ob01812d. [PMID: 34755753] - Lorain Geenen, Julie Nonnekens, Mark Konijnenberg, Sarah Baatout, Marion De Jong, An Aerts. Overcoming nephrotoxicity in peptide receptor radionuclide therapy using [177Lu]Lu-DOTA-TATE for the treatment of neuroendocrine tumours.
Nuclear medicine and biology.
2021 Nov; 102-103(?):1-11. doi:
10.1016/j.nucmedbio.2021.06.006. [PMID: 34242948] - Daneng Li, Megan Minnix, Rebecca Allen, James Bading, Junie Chea, Patty Wong, Nicole Bowles, Erasmus Poku, John E Shively. Preclinical PET Imaging of NTSR-1-Positive Tumors with 64Cu- and 68Ga-DOTA-Neurotensin Analogs and Therapy with an 225Ac-DOTA-Neurotensin Analog.
Cancer biotherapy & radiopharmaceuticals.
2021 Oct; 36(8):651-661. doi:
10.1089/cbr.2020.3926. [PMID: 32822229] - Benedikt Klasen, Euy Sung Moon, Frank Rösch. AAZTA5-squaramide ester competing with DOTA-, DTPA- and CHX-A″-DTPA-analogues: Promising tool for 177Lu-labeling of monoclonal antibodies under mild conditions.
Nuclear medicine and biology.
2021 May; 96-97(?):80-93. doi:
10.1016/j.nucmedbio.2021.03.007. [PMID: 33839678] - Riikka Viitanen, Olli Moisio, Petteri Lankinen, Xiang-Guo Li, Mikko Koivumäki, Sami Suilamo, Tuula Tolvanen, Kirsi Taimen, Markku Mali, Ia Kohonen, Ilpo Koskivirta, Vesa Oikonen, Helena Virtanen, Kristiina Santalahti, Anu Autio, Antti Saraste, Laura Pirilä, Pirjo Nuutila, Juhani Knuuti, Sirpa Jalkanen, Anne Roivainen. First-in-Humans Study of 68Ga-DOTA-Siglec-9, a PET Ligand Targeting Vascular Adhesion Protein 1.
Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
2021 04; 62(4):577-583. doi:
10.2967/jnumed.120.250696. [PMID: 32817143] - Anna Maria Trotta, Michela Aurilio, Crescenzo D'Alterio, Caterina Ieranò, Daria Di Martino, Antonio Barbieri, Antonio Luciano, Paolo Gaballo, Sara Santagata, Luigi Portella, Stefano Tomassi, Luciana Marinelli, Deborah Sementa, Ettore Novellino, Secondo Lastoria, Stefania Scala, Margret Schottelius, Salvatore Di Maro. Novel Peptide-Based PET Probe for Non-invasive Imaging of C-X-C Chemokine Receptor Type 4 (CXCR4) in Tumors.
Journal of medicinal chemistry.
2021 03; 64(6):3449-3461. doi:
10.1021/acs.jmedchem.1c00066. [PMID: 33660512] - Manuela Matesan, Darrell R Fisher, Roger Wong, Ajay K Gopal, Damian J Green, Brenda M Sandmaier, William Bensinger, John M Pagel, Johnnie Orozco, Oliver W Press, Ryan D Cassaday, Eric Hutchinson, Michelle Wanner, Sujit Pal, Carolyn Thostenson, Joseph G Rajendran. Biokinetics of Radiolabeled Monoclonal Antibody BC8: Differences in Biodistribution and Dosimetry Among Hematologic Malignancies.
Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
2020 09; 61(9):1300-1306. doi:
10.2967/jnumed.119.234443. [PMID: 32169919] - Aimi Zhang, Tianze Wu, Li Bian, Panli Li, Qiufang Liu, Dongjian Zhang, Qiaomei Jin, Jian Zhang, Gang Huang, Shaoli Song. Synthesis and Evaluation of Ga-68-Labeled Rhein for Early Assessment of Treatment-Induced Tumor Necrosis.
Molecular imaging and biology.
2020 06; 22(3):515-525. doi:
10.1007/s11307-019-01365-y. [PMID: 31250330] - Christof Rottenburger, Guillaume P Nicolas, Lisa McDougall, Felix Kaul, Michal Cachovan, A Hans Vija, Roger Schibli, Susanne Geistlich, Anne Schumann, Tilman Rau, Katharina Glatz, Martin Behe, Emanuel R Christ, Damian Wild. Cholecystokinin 2 Receptor Agonist 177Lu-PP-F11N for Radionuclide Therapy of Medullary Thyroid Carcinoma: Results of the Lumed Phase 0a Study.
Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
2020 04; 61(4):520-526. doi:
10.2967/jnumed.119.233031. [PMID: 31519804] - Benjamin Poret, Laurence Desrues, Marc-André Bonin, Martin Pédard, Martine Dubois, Richard Leduc, Romain Modzelewski, Pierre Decazes, Fabrice Morin, Pierre Vera, Hélène Castel, Pierre Bohn, Pierrick Gandolfo. Development of Novel 111-In-Labelled DOTA Urotensin II Analogues for Targeting the UT Receptor Overexpressed in Solid Tumours.
Biomolecules.
2020 03; 10(3):. doi:
10.3390/biom10030471. [PMID: 32204509] - Sarah M Cheal, Mitesh Patel, Guangbin Yang, Darren Veach, Hong Xu, Hong-Fen Guo, Pat B Zanzonico, Donald B Axworthy, Nai-Kong V Cheung, Ouathek Ouerfelli, Steven M Larson. An N-Acetylgalactosamino Dendron-Clearing Agent for High-Therapeutic-Index DOTA-Hapten Pretargeted Radioimmunotherapy.
Bioconjugate chemistry.
2020 03; 31(3):501-506. doi:
10.1021/acs.bioconjchem.9b00736. [PMID: 31891487] - Patty Wong, Lin Li, Junie Chea, Weidong Hu, Erasmus Poku, Todd Ebner, Nicole Bowles, Jeffrey Y C Wong, Paul J Yazaki, Stephen Sligar, John E Shively. Antibody Targeted PET Imaging of 64Cu-DOTA-Anti-CEA PEGylated Lipid Nanodiscs in CEA Positive Tumors.
Bioconjugate chemistry.
2020 03; 31(3):743-753. doi:
10.1021/acs.bioconjchem.9b00854. [PMID: 31961138] - Fei Li, Zhenzhong Zhang, Jiong Cai, Xi Chen, Ying Zhou, Xiangyi Ma, Qingjian Dong, Fang Li, Ling Xi. Primary Preclinical and Clinical Evaluation of 68Ga-DOTA-TMVP1 as a Novel VEGFR-3 PET Imaging Radiotracer in Gynecological Cancer.
Clinical cancer research : an official journal of the American Association for Cancer Research.
2020 03; 26(6):1318-1326. doi:
10.1158/1078-0432.ccr-19-1845. [PMID: 31843751] - Wenbo Wang, Frederikke P Fliedner, Anders E Hansen, Rasmus Eliasen, Fredrik Melander, Andreas Kjaer, Thomas L Andresen, Andreas I Jensen, Jonas R Henriksen. Preclinical evaluation of cationic DOTA-triarginine-lipid conjugates for theranostic liquid brachytherapy.
Nanotheranostics.
2020; 4(3):142-155. doi:
10.7150/ntno.44562. [PMID: 32483520] - Nazanin Pirooznia, Khosrou Abdi, Davood Beiki, Farshad Emami, Seyed Shahriar Arab, Omid Sabzevari, Zahra Pakdin-Parizi, Parham Geramifar. Radiosynthesis, Biological Evaluation, and Preclinical Study of a 68Ga-Labeled Cyclic RGD Peptide as an Early Diagnostic Agent for Overexpressed α v β 3 Integrin Receptors in Non-Small-Cell Lung Cancer.
Contrast media & molecular imaging.
2020; 2020(?):8421657. doi:
10.1155/2020/8421657. [PMID: 32292304] - Diane Reidy-Lagunes, Neeta Pandit-Taskar, Joseph A O'Donoghue, Simone Krebs, Kevin D Staton, Serge K Lyashchenko, Jason S Lewis, Nitya Raj, Mithat Gönen, Christian Lohrmann, Lisa Bodei, Wolfgang A Weber. Phase I Trial of Well-Differentiated Neuroendocrine Tumors (NETs) with Radiolabeled Somatostatin Antagonist 177Lu-Satoreotide Tetraxetan.
Clinical cancer research : an official journal of the American Association for Cancer Research.
2019 12; 25(23):6939-6947. doi:
10.1158/1078-0432.ccr-19-1026. [PMID: 31439583] - Mohini Guleria, Tapas Das, Jeyachitra Amirdhanayagam, Haladhar D Sarma, Ashutosh Dash. Preparation of [177Lu]Lu-DOTA-Ahx-Lys40-Exendin-4 for radiotherapy of insulinoma: a detailed insight into the radiochemical intricacies.
Nuclear medicine and biology.
2019 Nov; 78-79(?):31-40. doi:
10.1016/j.nucmedbio.2019.11.003. [PMID: 31731177] - Maximilian Klingler, Dominik Summer, Christine Rangger, Roland Haubner, Julie Foster, Jane Sosabowski, Clemens Decristoforo, Irene Virgolini, Elisabeth von Guggenberg. DOTA-MGS5, a New Cholecystokinin-2 Receptor-Targeting Peptide Analog with an Optimized Targeting Profile for Theranostic Use.
Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
2019 07; 60(7):1010-1016. doi:
10.2967/jnumed.118.221283. [PMID: 30530828] - Ambreen Khawar, Elisabeth Eppard, Frank Roesch, Hojjat Ahmadzadehfar, Stefan Kürpig, Michael Meisenheimer, Florian C Gaertner, Markus Essler, Ralph A Bundschuh. Preliminary results of biodistribution and dosimetric analysis of [68Ga]Ga-DOTAZOL: a new zoledronate-based bisphosphonate for PET/CT diagnosis of bone diseases.
Annals of nuclear medicine.
2019 Jun; 33(6):404-413. doi:
10.1007/s12149-019-01348-7. [PMID: 30877560] - Jie Zhang, Zi Wang, Huipan Liu, Liang Cai, Yue Feng, Ling Zhou, Hongyuan Wei, Ying Xie, Yue Chen. In vivo and in vitro evaluation of 177Lu-labeled DOTA-2-deoxy-D-glucose in mice. A novel radiopharmaceutical agent for cells imaging and therapy.
Hellenic journal of nuclear medicine.
2019 May; 22(2):103-110. doi:
10.1967/s002449911002. [PMID: 31273351] - Áron Roxin, Chengcheng Zhang, Sungjoon Huh, Mathieu Lepage, Zhengxing Zhang, Kuo-Shyan Lin, François Bénard, David M Perrin. A Metal-Free DOTA-Conjugated 18F-Labeled Radiotracer: [18F]DOTA-AMBF3-LLP2A for Imaging VLA-4 Over-Expression in Murine Melanoma with Improved Tumor Uptake and Greatly Enhanced Renal Clearance.
Bioconjugate chemistry.
2019 04; 30(4):1210-1219. doi:
10.1021/acs.bioconjchem.9b00146. [PMID: 30896929] - Rong Yuan, Fuchun Ge, Yong Liang, Yang Zhou, Limin Yang, Qiuquan Wang. Viruslike Element-Tagged Nanoparticle Inductively Coupled Plasma Mass Spectrometry Signal Multiplier: Membrane Biomarker Mediated Cell Counting.
Analytical chemistry.
2019 04; 91(8):4948-4952. doi:
10.1021/acs.analchem.9b00749. [PMID: 30938153] - John R Lever, Emily A Fergason-Cantrell, Terry L Carmack, Lisa D Watkinson, Fabio Gallazzi. Design, synthesis and evaluation of 111In labeled DOTA-conjugated tetrapeptides having high affinity and selectivity for mu opioid receptors.
Nuclear medicine and biology.
2019 03; 70(?):53-66. doi:
10.1016/j.nucmedbio.2019.02.001. [PMID: 30933866] - Michael W Linscheid. Molecules and elements for quantitative bioanalysis: The allure of using electrospray, MALDI, and ICP mass spectrometry side-by-side.
Mass spectrometry reviews.
2019 03; 38(2):169-186. doi:
10.1002/mas.21567. [PMID: 29603315] - Pardeep Kumar, Sushil K Tripathi, C P Chen, Eric Wickstrom, Mathew L Thakur. Evaluating Ga-68 Peptide Conjugates for Targeting VPAC Receptors: Stability and Pharmacokinetics.
Molecular imaging and biology.
2019 02; 21(1):130-139. doi:
10.1007/s11307-018-1207-x. [PMID: 29802552] - Sudipta Chakraborty, Dibakar Goswami, Rubel Chakravarty, Sahiralam Khan Mohammed, Haladhar Deb Sarma, Ashutosh Dash. Syntheses and evaluation of 68 Ga- and 153 Sm-labeled DOTA-conjugated bisphosphonate ligand for potential use in detection of skeletal metastases and management of pain arising from skeletal metastases.
Chemical biology & drug design.
2018 09; 92(3):1618-1626. doi:
10.1111/cbdd.13327. [PMID: 29729071] - Ermelinda Lucente, Hongguang Liu, Yang Liu, Xiang Hu, Enza Lacivita, Marcello Leopoldo, Zhen Cheng. Novel 64Cu Labeled RGD2-BBN Heterotrimers for PET Imaging of Prostate Cancer.
Bioconjugate chemistry.
2018 05; 29(5):1595-1604. doi:
10.1021/acs.bioconjchem.8b00113. [PMID: 29587479] - Sadaf Aghevlian, Yijie Lu, Mitchell A Winnik, David W Hedley, Raymond M Reilly. Panitumumab Modified with Metal-Chelating Polymers (MCP) Complexed to 111In and 177Lu-An EGFR-Targeted Theranostic for Pancreatic Cancer.
Molecular pharmaceutics.
2018 03; 15(3):1150-1159. doi:
10.1021/acs.molpharmaceut.7b01000. [PMID: 29314858] - Andreas I Jensen, Gregory W Severin, Anders E Hansen, Frederikke P Fliedner, Rasmus Eliasen, Ladan Parhamifar, Andreas Kjær, Thomas L Andresen, Jonas R Henriksen. Remote-loading of liposomes with manganese-52 and in vivo evaluation of the stabilities of 52Mn-DOTA and 64Cu-DOTA using radiolabelled liposomes and PET imaging.
Journal of controlled release : official journal of the Controlled Release Society.
2018 01; 269(?):100-109. doi:
10.1016/j.jconrel.2017.11.006. [PMID: 29122662] - Tilman Läppchen, Raffaella Rossin, Tiemen R van Mourik, Guillaume Gruntz, Freek J M Hoeben, Ron M Versteegen, Henk M Janssen, Johan Lub, Marc S Robillard. DOTA-tetrazine probes with modified linkers for tumor pretargeting.
Nuclear medicine and biology.
2017 Dec; 55(?):19-26. doi:
10.1016/j.nucmedbio.2017.09.001. [PMID: 29028502] - Mohamed Altai, Kristina Westerlund, Justin Velletta, Bogdan Mitran, Hadis Honarvar, Amelie Eriksson Karlström. Evaluation of affibody molecule-based PNA-mediated radionuclide pretargeting: Development of an optimized conjugation protocol and 177Lu labeling.
Nuclear medicine and biology.
2017 Nov; 54(?):1-9. doi:
10.1016/j.nucmedbio.2017.07.003. [PMID: 28810153] - Kazuma Ogawa, Atsushi Ishizaki, Kenichiro Takai, Yoji Kitamura, Akira Makino, Takashi Kozaka, Yasushi Kiyono, Kazuhiro Shiba, Akira Odani. Evaluation of Ga-DOTA-(D-Asp)n as bone imaging agents: D-aspartic acid peptides as carriers to bone.
Scientific reports.
2017 10; 7(1):13971. doi:
10.1038/s41598-017-14149-7. [PMID: 29070853] - Svend B Jensen, Meeri Käkelä, Lars Jødal, Olli Moisio, Aage K O Alstrup, Sirpa Jalkanen, Anne Roivainen. Exploring the radiosynthesis and in vitro characteristics of [68 Ga]Ga-DOTA-Siglec-9.
Journal of labelled compounds & radiopharmaceuticals.
2017 07; 60(9):439-449. doi:
10.1002/jlcr.3525. [PMID: 28556976] - Patty Wong, Lin Li, Junie Chea, Melissa K Delgado, Desiree Crow, Erasmus Poku, Barbara Szpikowska, Nicole Bowles, Divya Channappa, David Colcher, Jeffrey Y C Wong, John E Shively, Paul J Yazaki. PET imaging of 64Cu-DOTA-scFv-anti-PSMA lipid nanoparticles (LNPs): Enhanced tumor targeting over anti-PSMA scFv or untargeted LNPs.
Nuclear medicine and biology.
2017 Apr; 47(?):62-68. doi:
10.1016/j.nucmedbio.2017.01.004. [PMID: 28126683] - Junyong Dai, Miaode Wang, Hailong Liu. Highly selective enrichment of phosphopeptides using Zr4+-immobilized Titania nanoparticles.
Talanta.
2017 Mar; 164(?):222-227. doi:
10.1016/j.talanta.2016.11.058. [PMID: 28107921] - Nathalie M Grob, Martin Behe, Elisabeth von Guggenberg, Roger Schibli, Thomas L Mindt. Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates.
Journal of peptide science : an official publication of the European Peptide Society.
2017 Jan; 23(1):38-44. doi:
10.1002/psc.2948. [PMID: 28054429] - Giampiero Giovacchini, Elisabetta Giovannini, Mattia Riondato, Andrea Ciarmiello. Radiopharmaceuticals for the Diagnosis and Therapy of Neuroendocrine Differentiated Prostate Cancer.
Current radiopharmaceuticals.
2017; 10(1):6-15. doi:
10.2174/1874471009666161229123126. [PMID: 28034291] - Marian Meckel, Vojtěch Kubíček, Petr Hermann, Matthias Miederer, Frank Rösch. A DOTA based bisphosphonate with an albumin binding moiety for delayed body clearance for bone targeting.
Nuclear medicine and biology.
2016 Nov; 43(11):670-678. doi:
10.1016/j.nucmedbio.2016.07.009. [PMID: 27560354] - Masoumeh Zoghi, Amir R Jalilian, Ali Niazi, Fariba Johari-Daha, Behrouz Alirezapour, Saeed Ramezanpour. Development of a (68)Ga-peptide tracer for PET GnRH1-imaging.
Annals of nuclear medicine.
2016 Jul; 30(6):400-8. doi:
10.1007/s12149-016-1074-y. [PMID: 27083468] - Sangeeta Ray Banerjee, Zhengping Chen, Mrudula Pullambhatla, Ala Lisok, Jian Chen, Ronnie C Mease, Martin G Pomper. Preclinical Comparative Study of (68)Ga-Labeled DOTA, NOTA, and HBED-CC Chelated Radiotracers for Targeting PSMA.
Bioconjugate chemistry.
2016 Jun; 27(6):1447-55. doi:
10.1021/acs.bioconjchem.5b00679. [PMID: 27076393] - Simmyung Yook, Yijie Lu, Jenny Jooyoung Jeong, Zhongli Cai, Lemuel Tong, Ramina Alwarda, Jean-Philippe Pignol, Mitchell A Winnik, Raymond M Reilly. Stability and Biodistribution of Thiol-Functionalized and (177)Lu-Labeled Metal Chelating Polymers Bound to Gold Nanoparticles.
Biomacromolecules.
2016 Apr; 17(4):1292-302. doi:
10.1021/acs.biomac.5b01642. [PMID: 26974228] - R Kerdjoudj, M Pniok, C Alliot, V Kubíček, J Havlíčková, F Rösch, P Hermann, S Huclier-Markai. Scandium(III) complexes of monophosphorus acid DOTA analogues: a thermodynamic and radiolabelling study with (44)Sc from cyclotron and from a (44)Ti/(44)Sc generator.
Dalton transactions (Cambridge, England : 2003).
2016 Jan; 45(4):1398-409. doi:
10.1039/c5dt04084a. [PMID: 26675416] - Aanchal Ghai, Baljinder Singh, Puja Panwar Hazari, Michael K Schultz, Ambika Parmar, Pardeep Kumar, Sarika Sharma, Devinder Dhawan, Anil Kumar Mishra. Radiolabeling optimization and characterization of (68)Ga labeled DOTA-polyamido-amine dendrimer conjugate - Animal biodistribution and PET imaging results.
Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
2015 Nov; 105(?):40-46. doi:
10.1016/j.apradiso.2015.07.021. [PMID: 26232562] - Choong Mo Kang, Gwang Il An, Yearn Seong Choe. Hybrid lymph node imaging using 64Cu-labeled mannose-conjugated human serum albumin with and without indocyanine green.
Nuclear medicine communications.
2015 Oct; 36(10):1026-34. doi:
10.1097/mnm.0000000000000353. [PMID: 26068310] - Petra Kolenc Peitl, MariaLuisa Tamma, Marko Kroselj, Friederike Braun, Beatrice Waser, Jean Claude Reubi, Marija Sollner Dolenc, Helmut R Maecke, Rosalba Mansi. Stereochemistry of amino acid spacers determines the pharmacokinetics of (111)In-DOTA-minigastrin analogues for targeting the CCK2/gastrin receptor.
Bioconjugate chemistry.
2015 Jun; 26(6):1113-9. doi:
10.1021/acs.bioconjchem.5b00187. [PMID: 25971921] - Lorenzo Tei, Zsolt Baranyai, Luca Gaino, Attila Forgács, Adrienn Vágner, Mauro Botta. Thermodynamic stability, kinetic inertness and relaxometric properties of monoamide derivatives of lanthanide(III) DOTA complexes.
Dalton transactions (Cambridge, England : 2003).
2015 Mar; 44(12):5467-78. doi:
10.1039/c4dt03939d. [PMID: 25695351] - Yide He, Diego Esteban-Fernández, Michael W Linscheid. Novel approach for labeling of biopolymers with DOTA complexes using in situ click chemistry for quantification.
Talanta.
2015 Mar; 134(?):468-475. doi:
10.1016/j.talanta.2014.11.049. [PMID: 25618695] - Morten Persson, Dorthe Skovgaard, Malene Brandt-Larsen, Camilla Christensen, Jacob Madsen, Carsten H Nielsen, Tine Thurison, Thomas Levin Klausen, Søren Holm, Annika Loft, Anne Kiil Berthelsen, Michael Ploug, Helle Pappot, Klaus Brasso, Niels Kroman, Liselotte Højgaard, Andreas Kjaer. First-in-human uPAR PET: Imaging of Cancer Aggressiveness.
Theranostics.
2015; 5(12):1303-16. doi:
10.7150/thno.12956. [PMID: 26516369] - Pie Huda, Tina Binderup, Martin Cramer Pedersen, Søren Roi Midtgaard, Dennis Ringkjøbing Elema, Andreas Kjær, Mikael Jensen, Lise Arleth. PET/CT Based In Vivo Evaluation of 64Cu Labelled Nanodiscs in Tumor Bearing Mice.
PloS one.
2015; 10(7):e0129310. doi:
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